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Synthesis of atropisomerically defined, highly substituted biaryl scaffolds through catalytic enantioselective bromination and regioselective cross-coupling

  • Yale University

Research output: Contribution to journalArticlepeer-review

57 Scopus citations

Abstract

A selective sequence: An enantioselective synthesis (see scheme) of atropisomerically defined p-terphenyls, as well as tetra- and pentaaryl compounds is reported. The synthesis proceeds through sequential atropisomer-selective electrophilic aromatic substitution and regioselective palladium-catalyzed cross-coupling reactions.

Original languageEnglish
Pages (from-to)5125-5129
Number of pages5
JournalAngewandte Chemie - International Edition
Volume50
Issue number22
DOIs
StatePublished - May 23 2011

Keywords

  • atropisomerism
  • bromination
  • cross-coupling reactions
  • peptides
  • regioselectivity

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